Discovery and Optimization of Orally Bioavailable Phthalazone and Cinnolone Carboxylic Acid Derivatives as S1P2 Antagonists against Fibrotic Diseases
Author:
Affiliation:
1. Galapagos NV, Generaal De Wittelaan L11 A3, 2800 Mechelen, Belgium
2. Galapagos SASU, 102 avenue Gaston Roussel, 93230 Romainville, France
3. Fidelta Ltd., Prilaz Baruna Filipovića 29, ZagrebHR-10000, Croatia
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.1c01066
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