Structure–Affinity and Structure–Kinetic Relationship Studies of Benzodiazepine Derivatives for the Development of Efficacious Vasopressin V<sub>2</sub> Receptor Antagonists-Reference-Cited by-同舟云学术

Structure–Affinity and Structure–Kinetic Relationship Studies of Benzodiazepine Derivatives for the Development of Efficacious Vasopressin V₂ Receptor Antagonists

Published:2023-02-03 Issue:5 Volume:66 Page:3621-3634
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Cao Xudong¹,Wang Peng¹,Zhao Wenchao¹,Yuan Haoxing¹,Hu Hongtao¹,Chen Ting¹,Zhang Yixiao¹,Ren Ying¹,Su Limin¹,Fu Kequan¹,Liu Hongli¹,Guo Dong¹^ORCID

Affiliation:

1. Jiangsu Key Laboratory of New Drug Research and Clinical Pharmacy, Xuzhou Medical University, 209 Tongshan Road, Xuzhou, Jiangsu221004, China

Funder

Natural Science Foundation of Jiangsu Province

Major Basic Research Project of the Natural Science Foundation of the Jiangsu Higher Education Institutions

National Natural Science Foundation of China

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.3c00015

Reference27 articles.

1. Autosomal dominant polycystic kidney disease: Disrupted pathways and potential therapeutic interventions

2. Autosomal dominant polycystic kidney disease

3. Inhibition of renal cystic disease development and progression by a vasopressin V2 receptor antagonist

4. Effect of a Vasopressin V2 Receptor Antagonist on Polycystic Kidney Disease Development in a Rat Model

5. Pro: Tolvaptan delays the progression of autosomal dominant polycystic kidney disease

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