Superiority of the Triple-Acting 5-HT6R/5-HT3R Antagonist and MAO-B Reversible Inhibitor PZ-1922 over 5-HT6R Antagonist Intepirdine in Alleviation of Cognitive Deficits in Rats

Author:

Grychowska Katarzyna1ORCID,López-Sánchez Uriel2,Vitalis Mathieu3,Canet Geoffrey4,Satała Grzegorz5ORCID,Olejarz-Maciej Agnieszka1,Gołębiowska Joanna5,Kurczab Rafał5,Pietruś Wojciech5,Kubacka Monika1,Moreau Christophe2ORCID,Walczak Maria1ORCID,Blicharz-Futera Klaudia1ORCID,Bento Ophélie67,Bantreil Xavier6ORCID,Subra Gilles6ORCID,Bojarski Andrzej J.5ORCID,Lamaty Frédéric6,Becamel Carine7ORCID,Zussy Charleine3,Chaumont-Dubel Séverine7ORCID,Popik Piotr5ORCID,Nury Hugues2,Marin Philippe7ORCID,Givalois Laurent348,Zajdel Paweł1ORCID

Affiliation:

1. Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Str., 30-688 Kraków, Poland

2. Univ. Grenoble Alpes, CNRS, CEA, IBS, F-38000 Grenoble, France

3. Molecular Mechanisms in Neurodegenerative Dementia (MMDN) Laboratory, University of Montpellier, EPHE-PSL, INSERM U1198, 34-095 Montpellier, France

4. Faculty of Medicine, Laval University, CR-CHUQ, G1 V 4G2 Québec City (QC), Canada

5. Maj Institute of Pharmacology, Polish Academy of Sciences, 12 Smętna Str., 31-324 Kraków, Poland

6. IBMM, Université de Montpellier, CNRS, ENSCM, 34-293 Montpellier, France

7. Institut de Génomique Fonctionnelle, Université de Montpellier, CNRS, INSERM, 34-094 Montpellier, France

8. CNRS, 75-016 Paris, France

Funder

Agence Nationale de la Recherche

Université de Montpellier

Narodowe Centrum Nauki

Fondation pour la Recherche Médicale

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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