Selective Substrates and Activity-Based Probes for Imaging of the Human Constitutive 20S Proteasome in Cells and Blood Samples-Reference-Cited by-同舟云学术

Selective Substrates and Activity-Based Probes for Imaging of the Human Constitutive 20S Proteasome in Cells and Blood Samples

Published:2018-05-28 Issue:12 Volume:61 Page:5222-5234
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Rut Wioletta¹,Poręba Marcin¹²^ORCID,Kasperkiewicz Paulina¹²,Snipas Scott J.²,Drąg Marcin¹^ORCID

Affiliation:

1. Department of Bioorganic Chemistry, Faculty of Chemistry, Wroclaw University of Science and Technology, Wyb. Wyspianskiego 27, 50-370 Wroclaw, Poland

2. Program in Cell Death and Survival Networks, Sanford Burnham Prebys Medical Discovery Institute, La Jolla, California 92037, United States

Funder

Ministerstwo Nauki i Szkolnictwa Wyzszego

European Regional Development Fund

Narodowe Centrum Nauki

H2020 Marie Sklodowska-Curie Actions

Fundacja na rzecz Nauki Polskiej

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.8b00026

Reference52 articles.

1. The ubiquitin-proteasome pathway: on protein death and cell life

2. Drugging the undruggables: exploring the ubiquitin system for drug development

3. The 26S Proteasome: A Molecular Machine Designed for Controlled Proteolysis

4. The proteasome activator 11 S REG or PA28: chimeras implicate carboxyl-terminal sequences in oligomerization and proteasome binding but not in the activation of specific proteasome catalytic subunits 1 1Edited by W. Baumeister

5. Catalytic Activities of the 20 S Proteasome, a Multicatalytic Proteinase Complex

Cited by 28 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Structure-Guided Design and Synthesis of a Pyridazinone Series of Trypanosoma cruzi Proteasome Inhibitors;Journal of Medicinal Chemistry;2023-07-28

2. 20S proteasome hydrolysis of LLVY substrates to determine preferences for moieties in its primed substrate channel;Bioorganic & Medicinal Chemistry Letters;2023-04

3. Fluorescent Activity-Based Probe To Image and Inhibit Factor XIa Activity in Human Plasma;Journal of Medicinal Chemistry;2023-03-10

4. Synthetic peptide array on gold for the electrochemical assessment of the 20S proteasome activity and effect of inhibitory compounds;Applied Surface Science;2023-02

5. Diagnostic and therapeutic potential of protease inhibition;Molecular Aspects of Medicine;2022-12