Conjugation of Short Peptides to Dibenzodiazepinone-Type Muscarinic Acetylcholine Receptor Ligands Determines M2R Selectivity-Reference-Cited by-同舟云学术

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Conjugation of Short Peptides to Dibenzodiazepinone-Type Muscarinic Acetylcholine Receptor Ligands Determines M2R Selectivity

Published:2019-05-10 Issue:11 Volume:62 Page:5358-5369
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Pegoli Andrea¹,Wifling David¹,Gruber Corinna G.¹,She Xueke¹,Hübner Harald²,Bernhardt Günther¹^ORCID,Gmeiner Peter²^ORCID,Keller Max¹^ORCID

Affiliation:

1. Institute of Pharmacy, Faculty of Chemistry and Pharmacy, University of Regensburg, Universitätsstraße 31, D-93053 Regensburg, Germany

2. Department of Chemistry and Pharmacy, Medicinal Chemistry, Friedrich Alexander University, Nikolaus-Fiebiger-Straße 10, D-91058 Erlangen, Germany

Funder

Deutsche Forschungsgemeinschaft

China Scholarship Council

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.8b01967

Reference42 articles.

1. Overview of Muscarinic Receptor Subtypes

2. Allosteric Modulation of Muscarinic Acetylcholine Receptors

3. Crystal structures of the M1 and M4 muscarinic acetylcholine receptors

4. Therapeutic opportunities from muscarinic receptor research

5. Muscarinic M1receptor agonists and M2receptor antagonists as therapeutic targets in Alzheimer’s disease

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1. 8-[(4-benzylpiperazin-1-yl)methyl]-3-(2-chlorophenyl)-7-hydroxy-chromen-4-one is an activator of contractile activity of intestinal smooth muscles with reversible M2 cholinomimetic properties;Studia Biologica;2023-12

2. Stereochemistry-Driven Interactions of α,γ-Peptide Ligands with the Neuropeptide Y Y₄-Receptor;Journal of Medicinal Chemistry;2023-07-13

3. Designing drugs and chemical probes with the dualsteric approach;Chemical Society Reviews;2023

4. Click Chemistry-Enabled Conjugation Strategy for Producing Dibenzodiazepinone-Type Fluorescent Probes To Target M₂ Acetylcholine Receptors;Bioconjugate Chemistry;2022-11-03

5. N-Terminus to Arginine Side-Chain Cyclization of Linear Peptidic Neuropeptide Y Y4 Receptor Ligands Results in Picomolar Binding Constants;Journal of Medicinal Chemistry;2021-11-08

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