Design, Synthesis, and Biological Evaluation of 2-Nitroimidazopyrazin-one/-es with Antitubercular and Antiparasitic Activity-Reference-Cited by-同舟云学术

Design, Synthesis, and Biological Evaluation of 2-Nitroimidazopyrazin-one/-es with Antitubercular and Antiparasitic Activity

Published:2018-11-23 Issue:24 Volume:61 Page:11349-11371
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Jarrad Angie M.^ORCID,Ang Chee Wei,Debnath Anjan¹,Hahn Hye Jee¹,Woods Kyra²,Tan Lendl²,Sykes Melissa L.³,Jones Amy J.³,Pelingon Ruby,Butler Mark S.²^ORCID,Avery Vicky M.³,West Nicholas P.²,Karoli Tomislav^ORCID,Blaskovich Mark A. T.²^ORCID,Cooper Matthew A.²^ORCID

Affiliation:

1. Center for Discovery and Innovation in Parasitic Diseases, Skaggs School of Pharmacy and Pharmaceutical Sciences, University of California San Diego, La Jolla, California 92093, United States

2. Australian Infectious Diseases Research Centre, St. Lucia, Queensland 4067 Australia

3. Discovery Biology, Griffith Institute for Drug Discovery, Griffith University, Nathan, Queensland 4111, Australia

Funder

National Center for Advancing Translational Sciences

National Health and Medical Research Council

Australian Research Council

Wellcome Trust

Queensland Government

Institute for Molecular Bioscience, University of Queensland

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

http://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.8b01578

Reference59 articles.

1. Nitroimidazoles: Molecular Fireworks That Combat a Broad Spectrum of Infectious Diseases

2. A phase-3, double-blind, placebo-controlled study of the effectiveness and safety of single oral doses of secnidazole 2 g for the treatment of women with bacterial vaginosis

3. FDA Approves Symbiomix Therapeutics’ Solosec (Secnidazole) Oral Granules for the Treatment of Bacterial Vaginosis in Adult Women. https://symbiomix.com/fda-approves-symbiomix-therapeutics-solosec-secnidazole-oral-granules-treatment-bacterial-vaginosis-adult-women/ (accessed Sep 1, 2018).

4. Benznidazole approved for Chagas disease in children

5. Estimating and Mapping the Population at Risk of Sleeping Sickness

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