Design and Optimization of Sulfone Pyrrolidine Sulfonamide Antagonists of Transient Receptor Potential Vanilloid-4 with in Vivo Activity in a Pulmonary Edema Model-Reference-Cited by-同舟云学术

Design and Optimization of Sulfone Pyrrolidine Sulfonamide Antagonists of Transient Receptor Potential Vanilloid-4 with in Vivo Activity in a Pulmonary Edema Model

Published:2018-11-30 Issue:24 Volume:61 Page:11209-11220
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Pero Joseph E.^ORCID,Matthews Jay M.,Behm David J.,Brnardic Edward J.^ORCID,Brooks Carl,Budzik Brian W.,Costell Melissa H.,Donatelli Carla A.,Eisennagel Stephen H.,Erhard Karl,Fischer Michael C.,Holt Dennis A.,Jolivette Larry J.,Li Huijie,Li Peng,McAtee John J.,McCleland Brent W.,Pendrak Israil,Posobiec Lorraine M.,Rivera Katrina L.K.,Rivero Ralph A.,Roethke Theresa J.,Sender Matthew R.,Shu Arthur,Terrell Lamont R.,Vaidya Kalindi,Xu Xiaoping,Lawhorn Brian G.^ORCID

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.8b01344

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