Determination of Affinity and Residence Time of Potent Drug-Target Complexes by Label-free Biosensing
Author:
Affiliation:
1. Biophysical group, Biochemical and Cellular Pharmacology, Genentech, Inc., 1 DNA Way, South San Francisco, California 94080, United States
Funder
Genentech
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.7b01829
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4. Residence Time of Receptor−Ligand Complexes and Its Effect on Biological Function
5. The drug–target residence time model: a 10-year retrospective
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