1,2,4-Triazolo-[1,5-a]pyridine HIF Prolylhydroxylase Domain-1 (PHD-1) Inhibitors With a Novel Monodentate Binding Interaction
Author:
Affiliation:
1. Department of Computational Sciences and Crystallography, Takeda California Inc., 10410 Science Center Dr., San Diego, California 92121, United States
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.7b00352
Reference50 articles.
1. Regulation of theDrosophilabHLH-PAS Protein Sima by Hypoxia: Functional Evidence for Homology with Mammalian HIF-1α
2. Inducible operation of the erythropoietin 3' enhancer in multiple cell lines: evidence for a widespread oxygen-sensing mechanism.
3. A nuclear factor induced by hypoxia via de novo protein synthesis binds to the human erythropoietin gene enhancer at a site required for transcriptional activation.
4. Cellular and developmental control of O2 homeostasis by hypoxia-inducible factor 1α
5. Transcription Factor HIF-1 Is a Necessary Mediator of the Pasteur Effect in Mammalian Cells
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