Discovery, Development, and Cellular Delivery of Potent and Selective Bicyclic Peptide Inhibitors of Grb7 Cancer Target-Reference-Cited by-同舟云学术

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Discovery, Development, and Cellular Delivery of Potent and Selective Bicyclic Peptide Inhibitors of Grb7 Cancer Target

Published:2017-11-10 Issue:22 Volume:60 Page:9349-9359
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Watson Gabrielle M.¹,Kulkarni Ketav¹,Sang Jianrong¹²,Ma Xiuquan¹,Gunzburg Menachem J.¹,Perlmutter Patrick³,Wilce Matthew C.J.¹,Wilce Jacqueline A.¹^ORCID

Affiliation:

1. Biomedicine Discovery Institute, Department of Biochemistry and Molecular Biology, Monash University, Wellington Road, Clayton, VIC 3800, Australia

2. Department of Physiology, School of Medicine, Jiangsu University, Zhenjiang, Jiangsu 212013, P.R. China

3. School of Chemistry, Monash University, Wellington Road, Clayton, VIC 3800, Australia

Funder

National Health and Medical Research Council

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.7b01320

Reference48 articles.

1. Targeting protein–protein interactions as an anticancer strategy

2. Specificity in Signal Transduction

3. Hallmarks of Cancer: The Next Generation

4. Targeting protein−protein interfaces using macrocyclic peptides

5. The SH2 domain protein GRB-7 is co-amplified, overexpressed and in a tight complex with HER2 in breast cancer.

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1. Macrocycles and macrocyclization in anticancer drug discovery: Important pieces of the puzzle;European Journal of Medicinal Chemistry;2024-03

2. Membrane Permeability in a Large Macrocyclic Peptide Driven by a Saddle-Shaped Conformation;Journal of the American Chemical Society;2024-02-08

3. Grb7 knockout mice develop normally but litters born to knockout females fail to thrive;Developmental Dynamics;2023-12-23

4. Detecting Human Epidermal Growth Factor Receptor 2 (HER2) Amplification: Proof of Concept of an Alternative Approach;Cureus;2023-09-06

5. Grb7 knockout mice develop normally but litters born to knockout females fail to thrive;2023-07-01

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