Rapid Elaboration of Fragments into Leads by X-ray Crystallographic Screening of Parallel Chemical Libraries (REFiLX)

Author:

Bentley Matthew R.1,Ilyichova Olga V.1,Wang Geqing2,Williams Martin L.1,Sharma Gaurav1,Alwan Wesam S.1,Whitehouse Rebecca L.1,Mohanty Biswaranjan13,Scammells Peter J.1ORCID,Heras Begoña2,Martin Jennifer L.45,Totsika Makrina6,Capuano Ben13ORCID,Doak Bradley C.137,Scanlon Martin J.137ORCID

Affiliation:

1. Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University, 381 Royal Parade, Parkville, VIC 3052, Australia

2. Department of Biochemistry and Genetics, La Trobe Institute for Molecular Science, La Trobe University, Melbourne, VIC 3086, Australia

3. ARC Training Centre for Fragment Based Design, Monash Institute of Pharmaceutical Sciences, Monash University, 381 Royal Parade, Parkville, VIC 3052, Australia

4. Griffith Institute for Drug Discovery, Building N75, Brisbane Innovation Park, Don Young Road, Nathan, QLD 4111, Australia

5. Vice-Chancellor’s Unit, University of Wollongong, Northfields Avenue, Wollongong, NSW 2522, Australia

6. School of Biomedical Sciences, Institute of Health and Biomedical Innovation, Queensland University of Technology, Brisbane, QLD 4059, Australia

7. Monash Fragment Platform, Monash Institute of Pharmaceutical Sciences, Monash University, 381 Royal Parade, Parkville, VIC 3052, Australia

Funder

Monash University

National Health and Medical Research Council

Queensland University of Technology

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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