Nitrogen-Walk Approach to Explore Bioisosteric Replacements in a Series of Potent A2B Adenosine Receptor Antagonists-Reference-Cited by-同舟云学术

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Nitrogen-Walk Approach to Explore Bioisosteric Replacements in a Series of Potent A2B Adenosine Receptor Antagonists

Published:2020-06-23 Issue:14 Volume:63 Page:7721-7739
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Mallo-Abreu Ana,Prieto-Díaz Rubén,Jespers Willem¹^ORCID,Azuaje Jhonny,Majellaro Maria,Velando Carmen,García-Mera Xerardo,Caamaño Olga,Brea José²,Loza María I.²,Gutiérrez-de-Terán Hugo¹^ORCID,Sotelo Eddy^ORCID

Affiliation:

1. Department of Cell and Molecular Biology, Uppsala University, Uppsala SE 75124, Sweden

2. Centro Singular de Investigación en Medicina Molecular y Enfermedades Crónicas (CIMUS), Universidade de Santiago de Compostela, 15782 Santiago de Compostela, Spain

Funder

Vetenskapsr?det

Uppsala Universitet

Forskningsr?det om H?lsa, Arbetsliv och V?lf?rd

European Regional Development Fund

Lunds Universitet

European Cooperation in Science and Technology

Ume? Universitet

Conseller?a de Cultura, Educaci?n e Ordenaci?n Universitaria, Xunta de Galicia

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.0c00564

Reference76 articles.

1. International Union of Basic and Clinical Pharmacology. LXXXI. Nomenclature and Classification of Adenosine Receptors—An Update

2. Adenosine, an endogenous distress signal, modulates tissue damage and repair

3. Adenosine Receptors

4. Targeting immunosuppressive adenosine in cancer

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