Optimization of Acetazolamide-Based Scaffold as Potent Inhibitors of Vancomycin-Resistant Enterococcus-Reference-Cited by-同舟云学术

Optimization of Acetazolamide-Based Scaffold as Potent Inhibitors of Vancomycin-Resistant Enterococcus

Published:2020-07-28 Issue:17 Volume:63 Page:9540-9562
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Kaur Jatinder¹^ORCID,Cao Xufeng¹,Abutaleb Nader S.²^ORCID,Elkashif Ahmed²,Graboski Amanda L.¹,Krabill Aaron D.¹,AbdelKhalek Ahmed Hassan²^ORCID,An Weiwei¹,Bhardwaj Atul¹,Seleem Mohamed N.²³⁴^ORCID,Flaherty Daniel P.¹³⁴^ORCID

Affiliation:

1. Department of Medicinal Chemistry and Molecular Pharmacology, College of Pharmacy, Purdue University, 575 Stadium Mall Drive, West Lafayette, Indiana 47907, United States

2. Department of Comparative Pathobiology, College of Veterinary Medicine, Purdue University, 625 Harrison Street, West Lafayette, Indiana 47907, United States

3. Purdue Institute for Drug Discovery, 720 Clinic Drive, West Lafayette, Indiana 47907, United States

4. Purdue Institute of Inflammation, Immunology and Infectious Disease, 207 South Martin Jischke Drive, West Lafayette, Indiana 47907, United States

Funder

National Institute of Allergy and Infectious Diseases

Purdue Institute for Drug Discovery, Purdue University

Purdue College of Pharmacy, Purdue University

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.0c00734

Reference103 articles.

1. Antimicrobial-Resistant Pathogens Associated with Healthcare-Associated Infections Summary of Data Reported to the National Healthcare Safety Network at the Centers for Disease Control and Prevention, 2009–2010

2. Update on the antibiotic resistance crisis

3. Effect of Continuous and Sequential Therapy among Veterans Receiving Daptomycin or Linezolid for Vancomycin-Resistant Enterococcus faecium Bacteremia

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