A Novel N-Substituted Valine Derivative with Unique Peroxisome Proliferator-Activated Receptor γ Binding Properties and Biological Activities

Author:

Peiretti Franck1ORCID,Montanari Roberta2,Capelli Davide2,Bonardo Bernadette1,Colson Cécilia3,Amri Ez-Zoubir3,Grimaldi Marina4,Balaguer Patrick4,Ito Keiichi5,Roeder Robert G.5,Pochetti Giorgio2ORCID,Brunel Jean Michel6ORCID

Affiliation:

1. Aix Marseille University, INSERM, INRAE, C2VN, 13385 Marseille, France

2. Istituto di Cristallografia, Consiglio Nazionale delle Ricerche, Via Salaria km. 29.300, Monterotondo Stazione, 00015 Rome, Italy

3. Université Côte d’Azur, CNRS, Inserm, iBV, 06108 Nice, France

4. Institut de Recherche en Cancérologie de Montpellier (IRCM), INSERM, University of Montpellier, ICM, 34298 Montpellier, France

5. Laboratory of Biochemistry and Molecular Biology, The Rockefeller University, New York, New York 10065, United States

6. Aix Marseille University, INSERM, SSA, MCT, 13385 Marseille, France

Funder

Agence Nationale de la Recherche

Institut National de la Sant? et de la Recherche M?dicale

Aix-Marseille Universit?

Centre National de la Recherche Scientifique

National Institutes of Health

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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