Raloxifene-driven benzothiophene derivatives: Discovery, structural refinement, and biological evaluation as potent PPARγ modulators based on drug repurposing-Reference-Cited by-同舟云学术

Raloxifene-driven benzothiophene derivatives: Discovery, structural refinement, and biological evaluation as potent PPARγ modulators based on drug repurposing

Published:2024-04 Issue: Volume:269 Page:116325
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Liu Qingmei,Ma Lei,Chen Fangyuan,Zhang Shuyun,Huang Zexin,Zheng Xiufen,Chen Zikai,Ye Junwei,Hou Ning,Yi Wei^ORCID,Zhou Zhi

Funder

National Natural Science Foundation of China

Publisher

Elsevier BV

Reference65 articles.

1. Management of hyperglycaemia in type 2 diabetes, 2022. A consensus report by the American diabetes association (ADA) and the European association for the study of diabetes (EASD);Davies;Diabetes Care,2022

2. Type 2 diabetes: a multifaceted disease;Pearson;Diabetologia,2019

3. Type 2 diabetes mellitus, insulin resistance, and vitamin D;Sacerdote;Curr. Diabetes Rep.,2019

4. Pathophysiology of type 2 diabetes mellitus;Galicia-Garcia;Int. J. Mol. Sci.,2020

5. Macrovascular complications of Type 2 diabetes mellitus;Viigimaa;Curr. Vasc. Pharmacol.,2022

Cited by 2 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. An Overview of the Pharmacological Activities and Synthesis of Benzothiophene Derivatives;Medicinal Chemistry;2024-11

2. Structure-based screening, optimization and biological evaluation of novel chrysin-based derivatives as selective PPARγ modulators for the treatment of T2DM and hepatic steatosis;European Journal of Medicinal Chemistry;2024-10