Discovery of a Napabucasin PROTAC as an Effective Degrader of the E3 Ligase ZFP91-Reference-Cited by-同舟云学术

Discovery of a Napabucasin PROTAC as an Effective Degrader of the E3 Ligase ZFP91

Published:2021-01-28 Issue:3 Volume:64 Page:1626-1648
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Hanafi Maha¹²^ORCID,Chen Xinde¹,Neamati Nouri¹^ORCID

Affiliation:

1. Department of Medicinal Chemistry, College of Pharmacy and the Rogel Cancer Center, North Campus Research Complex, 1600 Huron Parkway, University of Michigan, Ann Arbor, Michigan 48109, United States

2. Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Cairo University, Cairo 11562, Egypt

Funder

National Cancer Institute

Ministry of Higher Education and Scientific Research

Forbes Institute for Cancer Discovery, University of Michigan

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.0c01897

Reference61 articles.

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5. Nucleus-Targeted, Echogenic Polymersomes for Delivering a Cancer Stemness Inhibitor to Pancreatic Cancer Cells

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