1. Centre
National de la Recherche Scientifique (CNRS), Centre de Recherche
en Cancérologie de Marseille (CRCM), UMR 7258; INSERM U1068; Institut Paoli-Calmettes; Aix-Marseille Université, UM105, 13273 Marseille, France
2. Department
of Organic Chemistry, Lobachevsky State University of Nizhni Novgorod, Gagarina av. 23, Nizhni Novgorod 603950, Russia
3. Screening
Platform AD2P, CNRS, AFMB UMR 7257, Aix-Marseille Université, 13288 Marseille, France
4. Cisbio Bioassays, R&D, Parc Marcel Boiteux, BP 84175, 30200 Codolet, France
5. Target
Discovery Institute, University of Oxford, NDM Research Building, Roosevelt
Drive, Oxford OX3 7FZ, U.K.
6. Structural
Genomics Consortium, University of Oxford, Old Road Campus Research Building,
Roosevelt Drive, Oxford OX3 7DQ, U.K.
7. Goethe-University, Institute for Pharmaceutical Chemistry and Buchmann
Institute for Life Science, Campus Riedberg, Max-von Laue Str. 9, 60438 Frankfurt am Main, Germany