Progress in the Development and Application of Small Molecule Inhibitors of Bromodomain–Acetyl-lysine Interactions-Reference-Cited by-同舟云学术

Progress in the Development and Application of Small Molecule Inhibitors of Bromodomain–Acetyl-lysine Interactions

Published:2012-09-27 Issue:22 Volume:55 Page:9393-9413
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Hewings David S.¹²,Rooney Timothy P. C.¹²,Jennings Laura E.¹²,Hay Duncan A.¹²,Schofield Christopher J.¹,Brennan Paul E.²,Knapp Stefan²,Conway Stuart J.¹

Affiliation:

1. Chemistry Research Laboratory, Department of Chemistry, University of Oxford, Mansfield Road, Oxford, OX1 3TA, U.K.

2. Nuffield Department of Clinical Medicine, Structural Genomics Consortium, University of Oxford, Old Road Campus Research Building, Roosevelt Drive, Oxford, OX3 7DQ, U.K.

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm300915b

Reference88 articles.

1. Acetylation: a regulatory modification to rival phosphorylation?

2. Lysine Acetylation Targets Protein Complexes and Co-Regulates Major Cellular Functions

3. Proteome-Wide Mapping of the Drosophila Acetylome Demonstrates a High Degree of Conservation of Lysine Acetylation

4. ACETYLATION AND METHYLATION OF HISTONES AND THEIR POSSIBLE ROLE IN THE REGULATION OF RNA SYNTHESIS

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