Discovery of Novel Inhibitor Scaffolds against the Metallo-β-lactamase VIM-2 by Surface Plasmon Resonance (SPR) Based Fragment Screening-Reference-Cited by-同舟云学术

Discovery of Novel Inhibitor Scaffolds against the Metallo-β-lactamase VIM-2 by Surface Plasmon Resonance (SPR) Based Fragment Screening

Published:2015-10-27 Issue:21 Volume:58 Page:8671-8682
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Christopeit Tony¹,Carlsen Trine Josefine O.¹,Helland Ronny¹,Leiros Hanna-Kirsti S.¹

Affiliation:

1. Department of Chemistry, Faculty of Science and Technology, The Norwegian Structural Biology Centre (NorStruct), UiT The Arctic University of Norway, N-9037 Tromsø, Norway

Funder

Norges Forskningsråd

Tromsø Research Foundation

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.5b01289

Reference40 articles.

1. Global Spread of Carbapenemase-producingEnterobacteriaceae

2. Carbapenemases: the Versatile β-Lactamases

3. Three Decades of β-Lactamase Inhibitors

4. 3-Mercapto-1,2,4-triazoles and N-acylated thiosemicarbazides as metallo-β-lactamase inhibitors

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