Investigation of (E)-3-[4-(2-Oxo-3-aryl-chromen-4-yl)oxyphenyl]acrylic Acids as Oral Selective Estrogen Receptor Down-Regulators-Reference-Cited by-同舟云学术

Investigation of (E)-3-[4-(2-Oxo-3-aryl-chromen-4-yl)oxyphenyl]acrylic Acids as Oral Selective Estrogen Receptor Down-Regulators

Published:2015-04-01 Issue:8 Volume:58 Page:3522-3533
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Degorce Sébastien L.¹²,Bailey Andrew¹,Callis Rowena³,De Savi Chris¹,Ducray Richard²,Lamont Gillian¹,MacFaul Philip¹,Maudet Mickael²,Martin Scott¹,Morgentin Rémy²,Norman Richard A.³,Peru Aurélien²,Pink Jennifer H.¹,Plé Patrick A.²,Roberts Bryan¹,Scott James S.¹

Affiliation:

1. Oncology Innovative Medicines Unit, AstraZeneca, Mereside, Alderley Park, Macclesfield, Cheshire SK10 4TG, United Kingdom

2. Oncology Innovative Medicines Unit, AstraZeneca, Centre de Recherches, Z.I. la Pompelle, BP1050, 51689 Reims Cedex 2, France

3. Discovery Sciences, AstraZeneca, Mereside, Alderley Park, Macclesfield, Cheshire SK10 4TG, United Kingdom

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.5b00066

Reference31 articles.

1. Selective oestrogen receptor modulation

2. Endocrinology and hormone therapy in breast cancer: Selective oestrogen receptor modulators and downregulators for breast cancer – have they lost their way?

3. Selective Estrogen Receptor Modulator Medicinal Chemistry At Merck. A Review

4. Contrasting Endocrine Activities of cis and trans Isomers in a Series of Substituted Triphenylethylenes

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