Novel Amino-pyrazole Ureas with Potent In Vitro and In Vivo Antileishmanial Activity-Reference-Cited by-同舟云学术

Novel Amino-pyrazole Ureas with Potent In Vitro and In Vivo Antileishmanial Activity

Published:2015-12-04 Issue:24 Volume:58 Page:9615-9624
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Mowbray Charles E.¹,Braillard Stéphanie¹,Speed William¹,Glossop Paul A.²,Whitlock Gavin A.²,Gibson Karl R.²,Mills James E. J.²,Brown Alan D.³,Gardner J. Mark F.⁴,Cao Yafeng⁵,Hua Wen⁵,Morgans Garreth L.⁶,Feijens Pim-Bart⁷,Matheeussen An⁷,Maes Louis J.⁷

Affiliation:

1. Drugs for Neglected Diseases initiative (DNDi), 15 Chemin Louis-Dunant, 1202 Geneva, Switzerland

2. Sandexis Medicinal Chemistry Ltd., Innovation House, Discovery Park, Ramsgate Road, Sandwich, Kent CT13 9ND, United Kingdom

3. Pfizer Worldwide Medicinal Chemistry, The Portway Building, Granta Park, Great Abington, Cambridge CB21 6GS, United Kingdom

4. AMG Consultants Ltd., Discovery Park House, Discovery Park, Ramsgate Road, Sandwich, Kent CT13 9ND, United Kingdom

5. WuXi AppTec (Wuhan) Company Ltd., 666 Gaoxin Road, East Lake High-Tech Development Zone, Wuhan 430075, People’s Republic of China

6. iThemba Pharmaceuticals, Building T5, Pinelands Site, High Street, Modderfontein 1609, Gauteng, South Africa

7. Laboratory for Microbiology, Parasitology and Hygiene (LMPH), University of Antwerp, S7, Universiteitsplein 1, 2610 Wilrijk, Antwerp, Belgium

Funder

Bundesministerium für Bildung und Forschung

Bill and Melinda Gates Foundation

Department for International Development

Ministerie van Buitenlandse Zaken

Direktion für Entwicklung und Zusammenarbeit

Médecins Sans Frontières

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.5b01456

Reference42 articles.

1. Fruitful Decade for Antileishmanial Compounds from 2002 to Late 2011

2. Visceral leishmaniasis treatment: What do we have, what do we need and how to deliver it?

3. WHO. Leishmaniasis.World Health Organ. Fact Sheet, 2014; Vol.375.

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