Click Chemistry in Lead Optimization of Boronic Acids as β-Lactamase Inhibitors-Reference-Cited by-同舟云学术

Click Chemistry in Lead Optimization of Boronic Acids as β-Lactamase Inhibitors

Published:2015-07-10 Issue:14 Volume:58 Page:5445-5458
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Caselli Emilia¹,Romagnoli Chiara¹,Vahabi Roza¹,Taracila Magdalena A.²,Bonomo Robert A.³²,Prati Fabio¹

Affiliation:

1. Department of Life Science, University of Modena and Reggio Emilia, via Campi 103, 41125 Modena, Italy

2. Departments of Medicine, Pharmacology, Biochemistry, and Molecular Biology and Microbiology, Case Western Reserve University, , Cleveland, Ohio 44106, United States

3. Research Service, Louis Stokes Cleveland Department of Veterans Affairs Medical Center, Cleveland, Ohio 44106, United States

Funder

National Institute of Allergy and Infectious Diseases

Harrington Discovery Institute, University Hospitals Case Medical Center

U.S. Department of Veterans Affairs

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.5b00341

Reference50 articles.

1. aWHO Library Cataloguing-in-Publication Data. Antimicrobial Resistance: Global Report on Surveillance 2014.www.who.int/drugresistance/documents/surveillancereport/en/(accessed April 2014).

2. The antibacterial lead discovery challenge

3. Confronting the challenges of discovery of novel antibacterial agents

4. Boron-containing inhibitors of synthetases

5. Not boring at all

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