Discovery and Optimization of Indoline-Based Compounds as Dual 5-LOX/sEH Inhibitors: In Vitro and In Vivo Anti-Inflammatory Characterization

Author:

Cerqua Ida1,Musella Simona2,Peltner Lukas Klaus3,D’Avino Danilo1ORCID,Di Sarno Veronica2,Granato Elisabetta1,Vestuto Vincenzo2,Di Matteo Rita1,Pace Simona3,Ciaglia Tania2,Bilancia Rossella13,Smaldone Gerardina2,Di Matteo Francesca2,Di Micco Simone4ORCID,Bifulco Giuseppe2ORCID,Pepe Giacomo2ORCID,Basilicata Manuela Giovanna2,Rodriquez Manuela2,Gomez-Monterrey Isabel M.1ORCID,Campiglia Pietro24ORCID,Ostacolo Carmine1ORCID,Roviezzo Fiorentina1,Werz Oliver3ORCID,Rossi Antonietta1,Bertamino Alessia2ORCID

Affiliation:

1. Department of Pharmacy, University Federico II of Naples, Via D. Montesano 49, 80131 Naples, Italy

2. Department of Pharmacy, University of Salerno, Via G. Paolo II 132, 84084 Fisciano, Salerno, Italy

3. Department of Pharmaceutical/Medicinal Chemistry, Institute of Pharmacy, Friedrich-Schiller-University, Philosophenweg 14, D-07743 Jena, Germany

4. European Biomedical Research Institute (EBRIS), Via S. De Renzi 50, 84125 Salerno, Italy

Funder

Freistaat Th?ringen

Associazione Italiana per la Ricerca sul Cancro

Universit? degli Studi di Napoli Federico II

European Social Fund

Regione Campania

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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