Exploring the Effect of Halogenation in a Series of Potent and Selective A2B Adenosine Receptor Antagonists

Author:

Prieto-Díaz Rubén123ORCID,González-Gómez Manuel12,Fojo-Carballo Hugo12,Azuaje Jhonny12,El Maatougui Abdelaziz12,Majellaro Maria12,Loza María I.45ORCID,Brea José45ORCID,Fernández-Dueñas Víctor67,Paleo M. Rita12ORCID,Díaz-Holguín Alejandro3,Garcia-Pinel Beatriz48ORCID,Mallo-Abreu Ana12ORCID,Estévez Juan C.12ORCID,Andújar-Arias Antonio12ORCID,García-Mera Xerardo2,Gomez-Tourino Iria4,Ciruela Francisco67ORCID,Salas Cristian O.9,Gutiérrez-de-Terán Hugo3ORCID,Sotelo Eddy12ORCID

Affiliation:

1. Center for Research in Biological Chemistry and Molecular Materials (CIQUS), University of Santiago de Compostela, 15782Santiago de Compostela, Spain

2. Department of Organic Chemistry, Faculty of Pharmacy, University of Santiago de Compostela, 15782Santiago de Compostela, Spain

3. Department of Cell and Molecular Biology, Uppsala University, Biomedical Center, 75124Uppsala, Sweden

4. Center for Research in Molecular Medicine and Chronic Diseases (CiMUS), University of Santiago de Compostela, 15782Santiago de Compostela, Spain

5. Department of Pharmacology, Pharmacy and Pharmaceutical Technology, Faculty of Pharmacy, University of Santiago de Compostela, 15782Santiago de Compostela, Spain

6. Pharmacology Unit, Department of Pathology and Experimental Therapeutics, Faculty of Medicine and Health Sciences, Institute of Neuroscience, University of Barcelona, 08907L’Hospitalet de Llobregat, Spain

7. Neuropharmacology and Pain Group, Neuroscience Program, Institut d’Investigació Biomèdica de Bellvitge, IDIBELL, 08907L’Hospitalet de Llobregat, Spain

8. Department of Biochemistry and Molecular Biology, Faculty of Pharmacy, University of Santiago de Compostela, 15782Santiago de Compostela, Spain

9. Department of Organic Chemistry, Faculty of Chemistry and Pharmacy, Pontificia Universidad Católica de Chile, Vicuña Mackenna 4860, Macul, Santiago7820436, Chile

Funder

Vetenskapsr?det

Forskningsr?det om H?lsa, Arbetsliv och V?lf?rd

Ministerio de Ciencia, Innovaci?n y Universidades

Agencia Estatal de Investigaci?n

Radiumhemmets Forskningsfonder

European Regional Development Fund

Xunta de Galicia

European Cooperation in Science and Technology

Cancerfonden

Conseller?a de Cultura, Educaci?n e Ordenaci?n Universitaria, Xunta de Galicia

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

同舟云学术

1.学者识别学者识别

2.学术分析学术分析

3.人才评估人才评估

"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370

www.globalauthorid.com

TOP

Copyright © 2019-2024 北京同舟云网络信息技术有限公司
京公网安备11010802033243号  京ICP备18003416号-3