Chemical Blockage of the Mitochondrial Rhomboid Protease PARL by Novel Ketoamide Inhibitors Reveals Its Role in PINK1/Parkin-Dependent Mitophagy

Author:

Poláchová Edita12,Bach Kathrin13,Heuten Elena45,Stanchev Stancho1,Tichá Anežka1,Lampe Philipp6,Majer Pavel1,Langer Thomas678,Lemberg Marius K.45,Stříšovský Kvido1ORCID

Affiliation:

1. Institute of Organic Chemistry and Biochemistry of the Czech Academy of Science, Flemingovo n. 2, Prague 160 00, Czech Republic

2. First Faculty of Medicine, Charles University, Kateřinská 32, Prague 121 08, Czech Republic

3. Department of Molecular Genetics, Faculty of Science, Charles University, Viničná 5, Prague 128 44, Czech Republic

4. Center for Molecular Biology of Heidelberg University (ZMBH), DKFZ-ZMBH Alliance, Im Neuenheimer Feld 282, Heidelberg 69120, Germany

5. Center for Biochemistry and Cologne Excellence Cluster on Cellular Stress Responses in Aging-Associated Diseases (CECAD), Medical Faculty, University of Cologne, Joseph-Stelzmann-Strasse 52, Cologne 50931, Germany

6. Institute for Genetics and Cologne Excellence Cluster on Cellular Stress Responses in Aging-Associated Diseases (CECAD), Medical Faculty, University of Cologne, Joseph-Stelzmann-Strasse 52, Cologne 50931, Germany

7. Center for Molecular Medicine (CMMC), Medical Faculty, University of Cologne, Joseph-Stelzmann-Strasse 52, Cologne 50931, Germany

8. Max-Planck-Institute for Biology of Ageing, Joseph-Stelzmann-Str. 9b, Cologne 50931, Germany

Funder

European Regional Development Fund

Ministerstvo ?kolstv?, Ml?de?e a Telov?chovy

Deutsche Forschungsgemeinschaft

Akademie Ved Cesk? Republiky

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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