Extensive targeting of chemical space at the prime side of ketoamide inhibitors of rhomboid proteases by branched substituents empowers their selectivity and potency-Reference-Cited by-同舟云学术

Extensive targeting of chemical space at the prime side of ketoamide inhibitors of rhomboid proteases by branched substituents empowers their selectivity and potency

Published:2024-09 Issue: Volume:275 Page:116606
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Bach Kathrin,Dohnálek Jan,Škerlová Jana,Kuzmík Ján,Poláchová Edita,Stanchev Stancho,Majer Pavel,Fanfrlík Jindřich,Pecina Adam,Řezáč Jan,Lepšík Martin,Borshchevskiy Valentin,Polovinkin Vitaly,Strisovsky Kvido^ORCID

Funder

Czech Science Foundation

Ministry of Education Youth and Sports of the Czech Republic

European Regional Development Fund

Publisher

Elsevier BV

Reference71 articles.

1. Rhomboid protease AarA mediates quorum-sensing in Providencia stuartii by activating TatA of the twin-arginine translocase;Stevenson;Proc. Natl. Acad. Sci. U.S.A.,2007

2. An Entamoeba histolytica rhomboid protease with atypical specificity cleaves a surface lectin involved in phagocytosis and immune evasion;Baxt;Genes Dev.,2008

3. Two Plasmodium rhomboid proteases preferentially cleave different adhesins implicated in all invasive stages of malaria;Baker;PLoS Pathog.,2006

4. Functional analysis of rhomboid proteases during Toxoplasma invasion;Shen;mBio,2014

5. Identification and characterization of a novel Aspergillus fumigatus rhomboid family putative protease, RbdA, involved in hypoxia sensing and virulence;Vaknin;Infect. Immun.,2016

Cited by 1 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Organizing Graphical User Interface tests from behavior‐driven development as videos to obtain stakeholders' feedback;Journal of Software: Evolution and Process;2024-08-05