Discovery of Novel Substrate-Competitive Lysine Methyltransferase G9a Inhibitors as Anticancer Agents-Reference-Cited by-同舟云学术

Discovery of Novel Substrate-Competitive Lysine Methyltransferase G9a Inhibitors as Anticancer Agents

Published:2023-03-08 Issue:6 Volume:66 Page:4059-4085
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Nishigaya Yosuke¹^ORCID,Takase Shohei²,Sumiya Tatsunobu¹,Kikuzato Ko,Sato Tomohiro^ORCID,Niwa Hideaki^ORCID,Sato Shin,Nakata Akiko,Sonoda Takeshi,Hashimoto Noriaki¹,Namie Ryosuke¹,Honma Teruki,Umehara Takashi^ORCID,Shirouzu Mikako,Koyama Hiroo,Yoshida Minoru³,Ito Akihiro²,Shirai Fumiyuki^ORCID

Affiliation:

1. Watarase Research Center, Discovery Research Headquarters, Kyorin Pharmaceutical Co. Ltd., 1848 Nogi, Shimotsuga-gun, Tochigi 329-0114, Japan

2. School of Life Sciences, Tokyo University of Pharmacy and Life Sciences, 1432-1 Horinouchi, Hachioji, Tokyo 192-0392, Japan

3. Department of Biotechnology, The University of Tokyo, 1-1-1 Yayoi, Bunkyo-ku, Tokyo 113-8657, Japan

Funder

RIKEN

Japan Agency for Medical Research and Development

Japan Society for the Promotion of Science

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine