Target-Focused Library Design by Pocket-Applied Computer Vision and Fragment Deep Generative Linking-Reference-Cited by-同舟云学术

Target-Focused Library Design by Pocket-Applied Computer Vision and Fragment Deep Generative Linking

Published:2022-10-18 Issue:20 Volume:65 Page:13771-13783
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Eguida Merveille¹^ORCID,Schmitt-Valencia Christel²,Hibert Marcel¹^ORCID,Villa Pascal²^ORCID,Rognan Didier¹^ORCID

Affiliation:

1. Laboratoire d’Innovation Thérapeutique, UMR7200 CNRS-Université de Strasbourg, F-67400Illkirch, France

2. Plateforme de Chimie Biologique Intégrative de Strasbourg, UAR3286 CNRS-Université de Strasbourg, Institut du Médicament de Strasbourg, F-67400Illkirch, France

Funder

Minist?re de l'Enseignement sup?rieur, de la Recherche et de l'Innovation

Universit? de Strasbourg

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.2c00931

Reference56 articles.

1. Twenty years on: the impact of fragments on drug discovery

2. Application of Fragment-Based Drug Discovery to Versatile Targets

3. Library Design Strategies To Accelerate Fragment‐Based Drug Discovery

4. Applied Biophysical Methods in Fragment-Based Drug Discovery

5. Fragment-Based Drug Discovery

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