Discovery and Structure-Based Design of Macrocyclic Peptides Targeting STUB1-Reference-Cited by-同舟云学术

Discovery and Structure-Based Design of Macrocyclic Peptides Targeting STUB1

Published:2022-07-19 Issue:14 Volume:65 Page:9789-9801
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Ng Simon¹^ORCID,Brueckner Alexander C.²^ORCID,Bahmanjah Soheila²,Deng Qiaolin²,Johnston Jennifer M.²^ORCID,Ge Lan³,Duggal Ruchia⁴,Habulihaz Bahanu⁵,Barlock Benjamin⁴,Ha Sookhee²,Sadruddin Ahmad¹,Yeo Constance¹,Strickland Corey²,Peier Andrea⁶^ORCID,Henry Brian¹,Sherer Edward C.²^ORCID,Partridge Anthony W.¹^ORCID

Affiliation:

1. Quantitative Biosciences, MSD, 8 Biomedical Grove, Singapore 138665

2. Computational & Structural Chemistry, Merck & Co., Inc., 2000 Galloping Hill Road, Kenilworth, New Jersey 07033, United States

3. Cell Sciences Innovation, Merck & Co., Inc., 2000 Galloping Hill Road, Kenilworth, New Jersey 07033, United States

4. ADME Group 2, Merck & Co., Inc., 33 Avenue Louis Pasteur, Boston, Massachusetts 02115, United States

5. PPDM ADME Transporters & In Vitro Technology, Merck & Co., Inc., 126 East Lincoln Ave, Rahway, New Jersey 07065, United States

6. Screening & Compound Profiling, Merck & Co., Inc., 2000 Galloping Hill Road, Kenilworth, New Jersey 07033, United States

Funder

Merck Sharp and Dohme

Merck

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.2c00406

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