Discovery of Potent OTUB1/USP8 Dual Inhibitors Targeting Proteostasis in Non-Small-Cell Lung Cancer

Author:

Tan Lingli12,Shan Hengyue23,Han Chao23ORCID,Zhang Zhenfeng4,Shen Jiali23,Zhang Xiao2,Xiang Huaijiang23,Lu Kuankuan23,Qi Chunting2,Li Ying2,Zhuang Guanglei4,Chen Gang1,Tan Li2ORCID

Affiliation:

1. School of Pharmacy, Fudan University, Shanghai 201203, China

2. Interdisciplinary Research Center on Biology and Chemistry, Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences, Shanghai 201210, China

3. University of Chinese Academy of Sciences, Beijing 100049, China

4. State Key Laboratory of Oncogenes and Related Genes, Shanghai Cancer Institute, Ren Ji Hospital, School of Medicine, Shanghai Jiao Tong University, Shanghai 200240, China

Funder

Shanghai Municipal Education Commission

Science and Technology Commission of Shanghai Municipality

National Natural Science Foundation of China

Chinese Academy of Sciences

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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