Potent, Efficacious, and Stable Cyclic Opioid Peptides with Long Lasting Antinociceptive Effect after Peripheral Administration-Reference-Cited by-同舟云学术

Potent, Efficacious, and Stable Cyclic Opioid Peptides with Long Lasting Antinociceptive Effect after Peripheral Administration

Published:2019-12-13 Issue:5 Volume:63 Page:2673-2687
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Stefanucci Azzurra¹^ORCID,Dimmito Marilisa Pia¹,Macedonio Giorgia¹,Ciarlo Laura²,Pieretti Stefano²^ORCID,Novellino Ettore³^ORCID,Lei Wei⁴,Barlow Deborah⁵,Houseknecht Karen L.⁵,Streicher John M.⁴^ORCID,Mollica Adriano¹^ORCID

Affiliation:

1. Dipartimento di Farmacia, Università di Chieti-Pescara “G. d’Annunzio”, Via dei Vestini 31, 66100 Chieti, Italy

2. Istituto Superiore di Sanità, Centro Nazionale Ricerca e Valutazione Preclinica e Clinica dei Farmaci, Viale Regina Elena 299, 00161 Rome, Italy

3. Dipartimento di Farmacia, Università di Napoli “Federico II”, Via D. Montesano, 49, 80131 Naples, Italy

4. Department of Pharmacology, College of Medicine, University of Arizona, Tucson, Arizona 85724, United States

5. Department of Biomedical Sciences, College of Osteopathic Medicine, University of New England, Biddeford, Maine 04005, United States

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.9b01963

Reference42 articles.

1. Pharmacologic Interventions for Pain Management

2. Structure-Activity Relationships of Biphalin Analogs and their Biological Evaluation on Opioid Receptors

3. Biphalin preferentially recruits peripheral opioid receptors to facilitate analgesia in a mouse model of cancer pain - A comparison with morphine

4. Antinociceptive profile of potent opioid peptide AM94, a fluorinated analogue of biphalin with non-hydrazine linker

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