Benzisothiazolinone Derivatives as Potent Allosteric Monoacylglycerol Lipase Inhibitors That Functionally Mimic Sulfenylation of Regulatory Cysteines-Reference-Cited by-同舟云学术

Benzisothiazolinone Derivatives as Potent Allosteric Monoacylglycerol Lipase Inhibitors That Functionally Mimic Sulfenylation of Regulatory Cysteines

Published:2019-11-12 Issue:3 Volume:63 Page:1261-1280
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Castelli Riccardo¹,Scalvini Laura¹^ORCID,Vacondio Federica¹²,Lodola Alessio¹^ORCID,Anselmi Mattia¹,Vezzosi Stefano¹,Carmi Caterina¹,Bassi Michele¹,Ferlenghi Francesca¹²,Rivara Silvia¹²^ORCID,Møller Ingvar R.³^ORCID,Rand Kasper D.³^ORCID,Daglian Jennifer,Wei Don,Dotsey Emmanuel Y.,Ahmed Faizy,Jung Kwang-Mook,Stella Nephi⁴^ORCID,Singh Simar⁴,Mor Marco¹²^ORCID,Piomelli Daniele

Affiliation:

1. Dipartimento di Scienze degli Alimenti e del Farmaco, Università degli Studi di Parma, Parco Area delle Scienze 27/A, I-43124 Parma, Italy

2. Centro Interdipartimentale Biopharmanet-tec, Università degli Studi di Parma, Parco Area delle Scienze, Tecnopolo Padiglione 33, I-43124 Parma, Italy

3. Department of Pharmacy, Universitetsparken 2, DK-2100 Copenhagen, Denmark

4. Department of Pharmacology, Psychiatry and Behavioral Sciences, University of Washington, Seattle, Washington 98195-7280, United States

Funder

Ministero dell???Istruzione, dell???Universit?? e della Ricerca

U.S. Department of Health and Human Services

Universit?? degli Studi di Parma and Fondazione Cariparma

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.9b01679