Characterization of the Binding Site of the Histamine H3 Receptor. 2. Synthesis, in Vitro Pharmacology, and QSAR of a Series of Monosubstituted Benzyl Analogues of Thioperamide-Reference-Cited by-同舟云学术

Characterization of the Binding Site of the Histamine H3 Receptor. 2. Synthesis, in Vitro Pharmacology, and QSAR of a Series of Monosubstituted Benzyl Analogues of Thioperamide

Published:2000-04-13 Issue:9 Volume:43 Page:1754-1761
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Windhorst Albert D.¹,Timmerman Henk¹,Worthington Edward A.¹,Bijloo Greetje J.¹,Nederkoorn Paul H. J.¹,Menge Wiro M. P. B.¹,Leurs Rob¹,Herscheid Jacobus D. M.¹

Affiliation:

1. Radionuclide Center, Vrije Universiteit, De Boelelaan 1085c, 1081 HV, Amsterdam, The Netherlands, and Leiden/Amsterdam Center for Drug Research (LACDR), Division of Medicinal Chemistry, Vrije Universiteit, De Boelelaan 1083, 1081 HV, Amsterdam, The Netherlands

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm981106w

Reference27 articles.

1. Molecular pharmacological aspects of histamine receptors

2. Three loci related to the src oncogene and tyrosine-specific protein kinase activity in Drosophila

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