Effects of rigidity on the selectivity of protein kinase inhibitors-Reference-Cited by-同舟云学术

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Effects of rigidity on the selectivity of protein kinase inhibitors

Published:2018-02 Issue: Volume:146 Page:519-528
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Assadieskandar Amir^ORCID,Yu Caiqun,Maisonneuve Pierre,Liu Xu,Chen Ying-Chu,Prakash G.K. Surya,Kurinov Igor,Sicheri Frank,Zhang Chao^ORCID

Funder

National Science Foundation

National Institute of Health

Canadian Cancer Society Research Institute

Canadian Institutes for Health Research

TD Bank postdoctoral fellowship

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference35 articles.

1. Protein kinase inhibitors: insights into drug design from structure;Noble;Science,2004

2. The ins and outs of selective kinase inhibitor development;Müller;Nat. Chem. Biol.,2015

3. Small-molecule kinase inhibitors: an analysis of FDA-approved drugs;Wu;Drug Discov. Today,2016

4. A small molecule–kinase interaction map for clinical kinase inhibitors;Fabian;Nat. Biotechnol.,2005

5. The selectivity of protein kinase inhibitors: a further update;Bain;Biochem. J.,2007

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5. Cytotoxic potential of three Sabal species grown in Egypt: a metabolomic and docking-based study;Natural Product Research;2020-11-28

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