Probing Binding Modes of Small Molecule Inhibitors to the Polo-Box Domain of Human Polo-like Kinase 1-Reference-Cited by-同舟云学术

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Probing Binding Modes of Small Molecule Inhibitors to the Polo-Box Domain of Human Polo-like Kinase 1

Published:2010-03-30 Issue:3 Volume:1 Page:110-114
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Liao Chenzhong¹,Park Jung-Eun²,Bang Jeong K.³,Nicklaus Marc C.¹,Lee Kyung S.²

Affiliation:

1. Chemical Biology Laboratory, Center for Cancer Research, National Cancer Institute, National Institutes of Health, Frederick, Maryland 21702

2. Laboratory of Metabolism, Center for Cancer Research, National Cancer Institute, National Institutes of Health, Bethesda, Maryland 20892

3. Korean Basic Science Institute, Ochang, Chung-Buk, 363-883, South Korea

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml100020e

Reference25 articles.

1. Polo-like kinases: conservation and divergence in their functions and regulation

2. Targeting polo-like kinase 1 for cancer therapy

3. A Genome-wide RNAi Screen Identifies Multiple Synthetic Lethal Interactions with the Ras Oncogene

4. A panel of isogenic human cancer cells suggests a therapeutic approach for cancers with inactivated p53

5. Pinning Down the Polo-Box Domain

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1. Leveraging the Fragment Molecular Orbital Method to Explore the PLK1 Kinase Binding Site and Polo-Box Domain for Potent Small-Molecule Drug Design;International Journal of Molecular Sciences;2023-10-27

2. Inhibitors of the PLK1 polo-box domain: drug design strategies and therapeutic opportunities in cancer;Expert Opinion on Drug Discovery;2023-01-01

3. Novel Macrocyclic Peptidomimetics Targeting the Polo-Box Domain of Polo-Like Kinase 1;Journal of Medicinal Chemistry;2022-01-14

4. Virtual screening of natural compounds as selective inhibitors of polo-like kinase-1 at C-terminal polo box and N-terminal catalytic domain;Journal of Biomolecular Structure and Dynamics;2021-10-20

5. Biological Activity of Purpurogallin and its Derivatives;Revista Virtual de Química;2021

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