Discovery of New Highly Potent Histamine H<sub>3</sub> Receptor Antagonists, Calcium Channel Blockers, and Acetylcholinesterase Inhibitors-Reference-Cited by-同舟云学术

Discovery of New Highly Potent Histamine H₃ Receptor Antagonists, Calcium Channel Blockers, and Acetylcholinesterase Inhibitors

Published:2024-08-29 Issue: Volume: Page:
ISSN:1948-7193
Container-title:ACS Chemical Neuroscience
language:en
Short-container-title:ACS Chem. Neurosci.

Author:

Malek Rim¹²,Sałat Kinga³^ORCID,Totoson Perle⁴,Karcz Tadeusz⁵,Refouvelet Bernard¹,Skrzypczak-Wiercioch Anna⁶,Maj Maciej⁷,Simakov Alexey⁴^ORCID,Martin Helene⁴,Siwek Agata⁸,Szałaj Natalia⁹,Godyń Justyna⁹^ORCID,Panek Dawid⁹,Więckowska Anna⁹^ORCID,Jozwiak Krzysztof⁷,Demougeot Celine⁴,Kieć-Kononowicz Katarzyna⁵,Chabchoub Fakher²,Iriepa Isabel¹⁰¹¹,Marco-Contelles José¹²¹³^ORCID,Ismaili Lhassane¹^ORCID

Affiliation:

1. Université de Franche-Comté, INSERM, UMR 1322 LINC, F-25000 Besançon, France

2. Laboratory of Applied Chemistry: Heterocycles, Lipids and Polymers, Faculty of Sciences of Sfax, University of Sfax, B. P 802, Sfax 3000, Tunisia

3. Department of Pharmacodynamics, Chair of Pharmacodynamics, Faculty of Pharmacy, Jagiellonian University Medical College, Kraków 30-688, Poland

4. Université de Franche-Comté, EFS, INSERM, UMR 1098 RIGHT, F-25000 Besançon, France

5. Department of Technology and Biotechnology of Drugs, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, Kraków 30-688, Poland

6. University Centre of Veterinary Medicine JU-UA, University of Agriculture in Krakow, 24/28 Mickiewicz St., Kraków 30-059, Poland

7. Department of Biopharmacy, Medical University of Lublin, ul. W. Chodzki 4a, Lublin 20-093, Poland

8. Department of Pharmacobiology, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, Kraków 30-688, Poland

9. Department of Physicochemical Drug Analysis, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, Kraków 30-688, Poland

10. Universidad de Alcalá. Departamento de Química Orgánica y Química Inorgánica, Alcalá de Henares, Madrid 28805, Spain

11. Instituto de Investigación Química Andrés M. del Río (IQAR), Universidad de Alcalá, Alcalá de Henares, Madrid 28805, Spain, Grupo DISCOBAC, Instituto de Investigación Sanitaria de Castilla-La Mancha (IDISCAM)

12. Laboratory of Medicinal Chemistry (IQOG, CSIC), C/ Juan de la Cierva 3, Madrid 28006, Spain

13. CIBER, ISCIII, Center for Biomedical Network Research on Rare Diseases (CIBERER), Madrid 28006, Spain

Funder

Ministry of Higher Education and Scientific Research

Minist?re de l'Europe et des Affaires ?trang?res

Conseil r?gional de Bourgogne-Franche-Comt?

Publisher

American Chemical Society (ACS)

Link

https://pubs.acs.org/doi/pdf/10.1021/acschemneuro.4c00341

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