Identification and Structure–Activity Relationship Study of Imidazo[1,2-a]pyridine-3-amines as First Selective Inhibitors of Excitatory Amino Acid Transporter Subtype 3 (EAAT3)-Reference-Cited by-同舟云学术

Identification and Structure–Activity Relationship Study of Imidazo[1,2-a]pyridine-3-amines as First Selective Inhibitors of Excitatory Amino Acid Transporter Subtype 3 (EAAT3)

Published:2019-10-01 Issue:10 Volume:10 Page:4414-4429
ISSN:1948-7193
Container-title:ACS Chemical Neuroscience
language:en
Short-container-title:ACS Chem. Neurosci.

Author:

Wu Peng¹^ORCID,Bjørn-Yoshimoto Walden E.¹,Staudt Markus¹,Jensen Anders A.¹,Bunch Lennart¹^ORCID

Affiliation:

1. Department of Drug Design and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Copenhagen DK-2100, Denmark

Funder

Sundhed og Sygdom, Det Frie Forskningsr?d

Lundbeckfonden

Publisher

American Chemical Society (ACS)

Subject

Cell Biology,Cognitive Neuroscience,Physiology,Biochemistry,General Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acschemneuro.9b00447

Reference53 articles.

1. Glutamate uptake

2. Excitatory amino acid transporters: recent insights into molecular mechanisms, novel modes of modulation and new therapeutic possibilities

3. SLC1 glutamate transporters

4. Excitatory amino acid transporters as potential drug targets

5. New views of glutamate transporter structure and function: Advances and challenges

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