Development of Novel δ Opioid Receptor Inverse Agonists without a Basic Nitrogen Atom and Their Antitussive Effects in Mice-Reference-Cited by-同舟云学术

Development of Novel δ Opioid Receptor Inverse Agonists without a Basic Nitrogen Atom and Their Antitussive Effects in Mice

Published:2019-08-09 Issue:9 Volume:10 Page:3939-3945
ISSN:1948-7193
Container-title:ACS Chemical Neuroscience
language:en
Short-container-title:ACS Chem. Neurosci.

Author:

Higashi Eika¹,Hirayama Shigeto¹²,Nikaido Jun³,Shibasaki Marie¹,Kono Tomomi¹,Honjo Ayaka¹,Ikeda Hiroko³,Kamei Junzo³⁴,Fujii Hideaki¹²^ORCID

Affiliation:

1. Laboratory of Medicinal Chemistry, School of Pharmacy, Kitasato University, 5-9-1, Shirokane, Minato-ku, Tokyo 108-8641, Japan

2. Medicinal Research Laboratories, School of Pharmacy, Kitasato University, 5-9-1, Shirokane, Minato-ku, Tokyo 108-8641, Japan

3. Department of Pathophysiology and Therapeutics, Hoshi University School of Pharmacy and Pharmaceutical Sciences, 2-4-41 Ebara, Shinagawa-ku, Tokyo 142-8501, Japan

4. Global Research Center for Innovative Life Science, Hoshi University School of Pharmacy and Pharmaceutical Sciences, 2-4-41 Ebara, Shinagawa-ku, Tokyo 142-8501, Japan

Publisher

American Chemical Society (ACS)

Subject

Cell Biology,Cognitive Neuroscience,Physiology,Biochemistry,General Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acschemneuro.9b00368

Reference39 articles.

1. Casy, A. F., and Parfitt, R. T. (1986) In Opioid Analgesics: Chemistry and Receptors, pp 9–104, Plenum Press, New York.

2. Design of peptidomimetic .delta. opioid receptor antagonists using the message-address concept

3. The most effective influence of 17-(3-ethoxypropyl) substituent on the binding affinity and the agonistic activity in KNT-127 derivatives, δ opioid receptor agonists

4. Novel Delta Opioid Receptor Agonists with Oxazatricyclodecane Structure

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