Design, Synthesis, and Characterization of the Macrocyclic Tetrapeptide cyclo[Pro-Sar-Phe-d-Phe]: A Mixed Opioid Receptor Agonist–Antagonist Following Oral Administration-Reference-Cited by-同舟云学术

Design, Synthesis, and Characterization of the Macrocyclic Tetrapeptide cyclo[Pro-Sar-Phe-d-Phe]: A Mixed Opioid Receptor Agonist–Antagonist Following Oral Administration

Published:2020-04-06 Issue:9 Volume:11 Page:1324-1336
ISSN:1948-7193
Container-title:ACS Chemical Neuroscience
language:en
Short-container-title:ACS Chem. Neurosci.

Author:

Ferracane Michael J.¹²,Brice-Tutt Ariana C.³,Coleman Jeremy S.¹,Simpson Grant G.¹,Wilson Lisa L.³,Eans Shainnel O.³,Stacy Heather M.³,Murray Thomas F.⁴,McLaughlin Jay P.³,Aldrich Jane V.¹^ORCID

Affiliation:

1. Department of Medicinal Chemistry, College of Pharmacy, University of Florida, Gainesville, Florida 32610, United States

2. Department of Chemistry, University of Redlands, Redlands, California 92373, United States

3. Department of Pharmacodynamics, College of Pharmacy, University of Florida, Gainesville, Florida 32610, United States

4. Department of Pharmacology, School of Medicine, Creighton University, Omaha, Nebraska 68178, United States

Funder

Office of the Secretary of Defense

National Institute on Drug Abuse

Publisher

American Chemical Society (ACS)

Subject

Cell Biology,Cognitive Neuroscience,Physiology,Biochemistry,General Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acschemneuro.0c00086

Reference52 articles.

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4. Psychotomimesis Mediated by κ Opiate Receptors

5. Assessment of the kappa opioid agonist, salvinorin A, as a punisher of drug self-administration in monkeys

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