Design, Synthesis, and Structure–Activity Relationship Exploration of Alkyl/Phenylalkyl Piperidine Analogues as Novel Highly Potent and Selective μ Opioid Receptor Agonists-Reference-Cited by-同舟云学术

Design, Synthesis, and Structure–Activity Relationship Exploration of Alkyl/Phenylalkyl Piperidine Analogues as Novel Highly Potent and Selective μ Opioid Receptor Agonists

Published:2020-08-27 Issue:2 Volume:12 Page:285-299
ISSN:1948-7193
Container-title:ACS Chemical Neuroscience
language:en
Short-container-title:ACS Chem. Neurosci.

Author:

Huang Huoming,Li Xinwei,Guo Wei,Zhu Chen,Qian Yuanyuan,Shen Qing,Xu Xuejun¹,Li Wei,Wang Yujun¹,Fu Wei^ORCID

Affiliation:

1. Shanghai Institute of Materia Medica, Chinese Academy of Science, Shanghai 201203, China

Funder

Youth Innovation Promotion Association of the Chinese Academy of Sciences

Shanghai Science and Technology Development Foundation

National Natural Science Foundation of China

Publisher

American Chemical Society (ACS)

Subject

Cell Biology,Cognitive Neuroscience,Physiology,Biochemistry,General Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acschemneuro.0c00487

Reference32 articles.

1. Opioid Complications and Side Effects

2. The Cost of Opioid-Related Adverse Drug Events

3. The µ Opioid Receptor and Ligands Acting at the µ Opioid Receptor, as Therapeutics and Potential Therapeutics

4. Opioid Pharmacology

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