Development of [Carbonyl-11C]AZ13198083, a Novel Histamine Type-3 Receptor Radioligand with Favorable Kinetics-Reference-Cited by-同舟云学术

Development of [Carbonyl-11C]AZ13198083, a Novel Histamine Type-3 Receptor Radioligand with Favorable Kinetics

Published:2018-01-23 Issue:5 Volume:9 Page:906-911
ISSN:1948-7193
Container-title:ACS Chemical Neuroscience
language:en
Short-container-title:ACS Chem. Neurosci.

Author:

Dahl Kenneth¹,Nakao Ryuji¹,Amini Nahid¹,Moein Mohammad Mahdi¹,Finnema Sjoerd¹,Malmquist Jonas²,Varnäs Katarina¹,Schou Magnus¹²^ORCID

Affiliation:

1. Department of Clinical Neuroscience, Center for Psychiatry Research, Karolinska Institutet and Stockholm County Council, SE-171 76 Stockholm, Sweden

2. PET Science Centre, Precision Medicine and Genomics, IMED Biotech Unit, AstraZeneca, Karolinska Institutet, S-171 76 Stockholm, Sweden

Funder

AstraZeneca

Publisher

American Chemical Society (ACS)

Subject

Cell Biology,Cognitive Neuroscience,Physiology,Biochemistry,General Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acschemneuro.7b00493

Reference35 articles.

1. Histamine H3 Receptor: A Potential Drug Target for the Treatment of Central Nervous System Disorders

2. The medicinal chemistry and therapeutic potentials of ligands of the histamine H3 receptor

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4. Characterization of histamine H3 receptors in Alzheimer's Disease brain and amyloid over-expressing TASTPM mice

5. Obesity: Current and potential pharmacotherapeutics and targets

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