Indanesulfonamides as Carbonic Anhydrase Inhibitors. Toward Structure-Based Design of Selective Inhibitors of the Tumor-Associated Isozyme CA IX-Reference-Cited by-同舟云学术

Indanesulfonamides as Carbonic Anhydrase Inhibitors. Toward Structure-Based Design of Selective Inhibitors of the Tumor-Associated Isozyme CA IX

Published:2006-04-01 Issue:9 Volume:49 Page:2743-2749
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Thiry Anne¹,Ledecq Marie¹,Cecchi Alessandro¹,Dogné Jean-Michel¹,Wouters Johan¹,Supuran Claudiu T.¹,Masereel Bernard¹

Affiliation:

1. Drug Design and Discovery Center, University of Namur, 61 rue de Bruxelles, 5000 Namur, Belgium, and Polo Scientifico, Laboratorio di Chimica Bioinorganica, Rm. 188, Università degli Studi di Firenze, Via della Lastruccia 3, 50019 Sesto Fiorentino, Florence, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm0600287

Reference47 articles.

1. Supuran, C. T. Carbonic Anhydrases: Catalytic and Inhibition Mechanisms, Distribution and Physiological Roles.Carbonic Anhyrdase.Its Inhibitors and Activators; CRC Press: London, 2004; pp 1−23.

2. Carbonic anhydrase inhibitors and their therapeutic potential

3. Carbonic Anhydrase

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