Investigation of 3-sulfamoyl coumarins against cancer-related IX and XII isoforms of human carbonic anhydrase as well as cancer cells leads to the discovery of 2-oxo-2H-benzo[h]chromene-3-sulfonamide – A new caspase-activating proapoptotic agent-Reference-Cited by-同舟云学术

Investigation of 3-sulfamoyl coumarins against cancer-related IX and XII isoforms of human carbonic anhydrase as well as cancer cells leads to the discovery of 2-oxo-2H-benzo[h]chromene-3-sulfonamide – A new caspase-activating proapoptotic agent

Published:2021-10 Issue: Volume:222 Page:113589
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Dar'in Dmitry,Kantin Grigory,Kalinin Stanislav,Sharonova Tatiana,Bunev Alexander^ORCID,Ostapenko Gennady I.,Nocentini Alessio^ORCID,Sharoyko Vladimir,Supuran Claudiu T.^ORCID,Krasavin Mikhail

Funder

Russian Foundation for Basic Research

Russian Science Foundation

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

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2. Coumarins as factor XIIa inhibitors: Potency and selectivity improvements using a fragment-based strategy;European Journal of Medicinal Chemistry;2023-11

3. Design, synthesis, and biological investigation of selective human carbonic anhydrase II, IX, and XII inhibitors using 7-aryl/heteroaryl triazolopyrimidines bearing a sulfanilamide scaffold;Journal of Enzyme Inhibition and Medicinal Chemistry;2023-10-18

4. Synthesis, biological evaluation and theoretical studies of ( E )-1-(4-sulfamoyl-phenylethyl)-3-arylidene-5-aryl-1H-pyrrol-2(3H)-ones as human carbonic anhydrase inhibitors;Journal of Enzyme Inhibition and Medicinal Chemistry;2023-03-23

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