Neoceptor Concept Based on Molecular Complementarity in GPCRs: A Mutant Adenosine A3 Receptor with Selectively Enhanced Affinity for Amine-Modified Nucleosides-Reference-Cited by-同舟云学术

Neoceptor Concept Based on Molecular Complementarity in GPCRs: A Mutant Adenosine A3 Receptor with Selectively Enhanced Affinity for Amine-Modified Nucleosides

Published:2001-10-16 Issue:24 Volume:44 Page:4125-4136
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Jacobson Kenneth A.¹,Gao Zhan-Guo¹,Chen Aishe¹,Barak Dov¹,Kim Soon-Ai¹,Lee Kyeong¹,Link Andreas¹,Rompaey Philippe Van¹,van Calenbergh Serge¹,Liang Bruce T.¹

Affiliation:

1. Molecular Recognition Section, Laboratory of Bioorganic Chemistry, National Institute of Diabetes and Digestive and Kidney Diseases, National Institutes of Health, Bethesda, Maryland 20892, Department of Medicine, Cardiovascular Division, and Department of Pharmacology, University of Pennsylvania Medical Center, Philadelphia, Pennsylvania 19104, Laboratorium voor Medicinale Chemie (FFW), Harelbekestraat 72, B-9000 Gent, Belgium, and Institut für Pharmazie, Fachbereich Chemie, Universität Hamburg,...

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm010232o

Reference57 articles.

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