Structural Analysis and Optimization of NK1 Receptor Antagonists through Modulation of Atropisomer Interconversion Properties-Reference-Cited by-同舟云学术

Structural Analysis and Optimization of NK1 Receptor Antagonists through Modulation of Atropisomer Interconversion Properties

Published:2003-12-23 Issue:3 Volume:47 Page:519-529
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Albert Jeffrey S.¹,Ohnmacht Cyrus¹,Bernstein Peter R.¹,Rumsey William L.¹,Aharony David¹,Alelyunas Yun¹,Russell Daniel J.¹,Potts William¹,Sherwood Scott A.¹,Shen Lihong¹,Dedinas Robert F.¹,Palmer William E.¹,Russell Keith¹

Affiliation:

1. CNS Discovery Research, AstraZeneca Pharmaceuticals LP, 1800 Concord Pike, P.O. Box 15437, Wilmington, Delaware 19850-5437, and EST, AstraZeneca Pharmaceuticals LP, Waltham, Massachusetts 02451

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm030197g

Reference48 articles.

1. Neurokinin1 Receptor Antagonists as Potential Antidepressants

2. Dual neurokinin NK1/NK2 receptor antagonists

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