Novel and Highly Potent 5-HT3 Receptor Agonists Based on a Pyrroloquinoxaline Structure-Reference-Cited by-同舟云学术

Novel and Highly Potent 5-HT3 Receptor Agonists Based on a Pyrroloquinoxaline Structure

Published:1997-10-01 Issue:22 Volume:40 Page:3670-3678
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Campiani Giuseppe¹,Cappelli Andrea¹,Nacci Vito¹,Anzini Maurizio¹,Vomero Salvatore¹,Hamon Michel¹,Cagnotto Alfredo¹,Fracasso Claudia¹,Uboldi Chiara¹,Caccia Silvio¹,Consolo Silvana¹,Mennini Tiziana¹

Affiliation:

1. Dipartimento Farmaco Chimico Tecnologico, Universitá di Siena, Banchi di Sotto 55, 53100 Siena, Italy, Neurobiologie Cellulaire et Functionnelle, Istitut National de la Santé et de la Recherche Medicale (INSERM) U.288, Faculté de Medicine Pitié-Salpetriere 91, boulevard del' Hopital, 75634 Paris, Cedex 13, France, and Istituto di Ricerche Farmacologiche “Mario Negri”, via Eritrea 62, 20127 Milano, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm970376w

Reference21 articles.

1. 5-HT3 receptors

2. Further studies on the blockade of 5-HT depolarizations of rabbit vagal afferent and sympathetic ganglion cells by MDL 72222 and other antagonists

3. Characteristics of [14C]Guanidinium Accumulation in NG 108-15 Cell Exposed to Serotonin 5-HT3Receptor Ligands and Substance P

4. Common pharmacological and physico-chemical properties of 5-HT3 binding sites in the rat cerebral cortex and NG 108-15 clonal cells

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