Optimization of the Central Core of Indolinone–Acetic Acid-Based CRTH2 (DP2) Receptor Antagonists-Reference-Cited by-同舟云学术

Optimization of the Central Core of Indolinone–Acetic Acid-Based CRTH2 (DP2) Receptor Antagonists

Published:2011-06-13 Issue:8 Volume:2 Page:644-649
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Crosignani Stefano¹,Jorand-Lebrun Catherine¹,Page Patrick¹,Campbell Gordon¹,Colovray Véronique¹,Missotten Marc¹,Humbert Yves¹,Cleva Christophe¹,Arrighi Jean-François¹,Gaudet Marilène¹,Johnson Zoe¹,Ferro Pamela¹,Chollet André¹

Affiliation:

1. Merck Serono S.A., 9 chemin des Mines, CH-1202 Geneva, Switzerland

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml2001196

Reference19 articles.

1. Antagonism of the prostaglandin D2 receptors DP1 and CRTH2 as an approach to treat allergic diseases

2. Prostaglandin D2 Selectively Induces Chemotaxis in T Helper Type 2 Cells, Eosinophils, and Basophils via Seven-Transmembrane Receptor Crth2

3. Prostaglandin D2-Induced Eosinophilic Airway Inflammation Is Mediated by CRTH2 Receptor

4. CRTH2 is the most reliable marker for the detection of circulating human type 2 Th and type 2 T cytotoxic cells in health and disease

5. Prostaglandin D2 Inhibits Airway Dendritic Cell Migration and Function in Steady State Conditions by Selective Activation of the D Prostanoid Receptor 1

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