Ligand Efficiency Driven Design of New Inhibitors of Mycobacterium tuberculosis Transcriptional Repressor EthR Using Fragment Growing, Merging, and Linking Approaches-Reference-Cited by-同舟云学术

Ligand Efficiency Driven Design of New Inhibitors of Mycobacterium tuberculosis Transcriptional Repressor EthR Using Fragment Growing, Merging, and Linking Approaches

Published:2014-05-28 Issue:11 Volume:57 Page:4876-4888
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Villemagne Baptiste¹²³⁴⁵,Flipo Marion¹²³⁴⁵,Blondiaux Nicolas¹³⁴⁵⁶,Crauste Céline¹²³⁴⁵,Malaquin Sandra¹²³⁴⁵,Leroux Florence¹²³⁴⁵,Piveteau Catherine¹²³⁴⁵,Villeret Vincent¹³⁷,Brodin Priscille¹³⁴⁶⁸,Villoutreix Bruno O.⁹¹⁰,Sperandio Olivier⁹¹⁰,Soror Sameh H.¹¹,Wohlkönig Alexandre¹¹,Wintjens René⁷¹²,Deprez Benoit¹²³⁴⁵,Baulard Alain R.¹³⁴⁵⁶,Willand Nicolas¹²³⁴⁵

Affiliation:

1. Université Lille Nord de France, F-59044 Lille, France

2. Biostructures and Drug Discovery, INSERM U761, F-59006 Lille, France

3. UDSL, F-59000 Lille, France

4. Institut Pasteur de Lille, F-59019 Lille, France

5. PRIM, F-59006 Lille, France

6. INSERM U1019, F-59019 Lille, France

7. IRI, USR 3078 CNRS, F-59658 Villeneuve d’Ascq, France

8. CNRS UMR8204, F-59021 Lille, France

9. INSERM, UMRS 973, MTi, F- 75013 Paris, France

10. Univ Paris Diderot, F-75205 Paris, France

11. Structural Biology Brussels and Molecular and Cellular Interactions, VIB, Brussels, Belgium