Potent and Selective Aurora Inhibitors Identified by the Expansion of a Novel Scaffold for Protein Kinase Inhibition-Reference-Cited by-同舟云学术

Potent and Selective Aurora Inhibitors Identified by the Expansion of a Novel Scaffold for Protein Kinase Inhibition

Published:2005-03-10 Issue:8 Volume:48 Page:3080-3084
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Fancelli Daniele¹,Berta Daniela¹,Bindi Simona¹,Cameron Alexander¹,Cappella Paolo¹,Carpinelli Patrizia¹,Catana Cornel¹,Forte Barbara¹,Giordano Patrizia¹,Giorgini Maria Laura¹,Mantegani Sergio¹,Marsiglio Aurelio¹,Meroni Maurizio¹,Moll Juergen¹,Pittalà Valeria¹,Roletto Fulvia¹,Severino Dino¹,Soncini Chiara¹,Storici Paola¹,Tonani Roberto¹,Varasi Mario¹,Vulpetti Anna¹,Vianello Paola¹

Affiliation:

1. Nerviano Medical Sciences - Oncology, via Pasteur 10, 20014 Nerviano, Milan, Italy

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm049076m

Reference14 articles.

1. Aurora kinases link chromosome segregation and cell division to cancer susceptibility

2. Dawn of Aurora kinase inhibitors as anticancer drugs

3. Aurora-C kinase is a novel chromosomal passenger protein that can complement Aurora-B kinase function in mitotic cells

4. A homologue of Drosophila aurora kinase is oncogenic and amplified in human colorectal cancers

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