Stromelysin Inhibitors Designed from Weakly Bound Fragments: Effects of Linking and Cooperativity
Author:
Affiliation:
1. Contribution from the Pharmaceutical Discovery Division, Abbott Laboratories, Abbott Park, Illinois 60064
Publisher
American Chemical Society (ACS)
Subject
Colloid and Surface Chemistry,Biochemistry,General Chemistry,Catalysis
Link
https://pubs.acs.org/doi/pdf/10.1021/ja9702780
Reference26 articles.
1. Discovery of Potent Nonpeptide Inhibitors of Stromelysin Using SAR by NMR
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3. On the attribution and additivity of binding energies
4. Janin, J.Proteins: Struct., Funct., Genet.1995,21, 30−39.
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